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    • Potent and subtype-selective dopamine D2 receptor biased partial agonists discovered via an Ugi-based approach 

      Mallo-Abreu, Ana; Reyes Resina, Irene; Azuaje Guerrero, Jhonny Alberto; Franco, Rafael; García Rey, Aitor; Majellaro, María; Miranda Pastoriza, Darío; García Mera, Xerardo Xusto; Jespers, Willem; Gutiérrez de Terán, Hugo; Navarro, Gemma; Sotelo, Eddy (ACS Publications, 2021)
      Using a previously unexplored, efficient, and versatile multicomponent method, we herein report the rapid generation of novel potent and subtype-selective DRD2 biased partial agonists. This strategy exemplifies the search ...





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